DE122011100044I1 - Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung. - Google Patents

Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung.

Info

Publication number
DE122011100044I1
DE122011100044I1 DE201112100044 DE122011100044C DE122011100044I1 DE 122011100044 I1 DE122011100044 I1 DE 122011100044I1 DE 201112100044 DE201112100044 DE 201112100044 DE 122011100044 C DE122011100044 C DE 122011100044C DE 122011100044 I1 DE122011100044 I1 DE 122011100044I1
Authority
DE
Germany
Prior art keywords
alkyl
radical
nhco
alkoxy
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE201112100044
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bausch Health US LLC
Original Assignee
Valeant Pharmaceuticals North America LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Valeant Pharmaceuticals North America LLC filed Critical Valeant Pharmaceuticals North America LLC
Publication of DE122011100044I1 publication Critical patent/DE122011100044I1/de
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/34Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C07C233/42Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • C07C233/43Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of a saturated carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/26Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring
    • C07C271/28Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atom of at least one of the carbamate groups bound to a carbon atom of a six-membered aromatic ring to a carbon atom of a non-condensed six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/28Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/40Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
DE201112100044 1992-01-08 2011-09-07 Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung. Pending DE122011100044I1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4200259A DE4200259A1 (de) 1992-01-08 1992-01-08 Neue 1,2,4-triaminobenzol-derivate und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
DE122011100044I1 true DE122011100044I1 (de) 2012-01-19

Family

ID=6449201

Family Applications (3)

Application Number Title Priority Date Filing Date
DE4200259A Withdrawn DE4200259A1 (de) 1992-01-08 1992-01-08 Neue 1,2,4-triaminobenzol-derivate und verfahren zu deren herstellung
DE59205496T Expired - Lifetime DE59205496D1 (de) 1992-01-08 1992-12-10 Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung
DE201112100044 Pending DE122011100044I1 (de) 1992-01-08 2011-09-07 Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
DE4200259A Withdrawn DE4200259A1 (de) 1992-01-08 1992-01-08 Neue 1,2,4-triaminobenzol-derivate und verfahren zu deren herstellung
DE59205496T Expired - Lifetime DE59205496D1 (de) 1992-01-08 1992-12-10 Neue 1,2,4-Triaminobenzol-Derivate und Verfahren zu deren Herstellung

Country Status (13)

Country Link
US (1) US5384330A (de)
EP (1) EP0554543B1 (de)
JP (1) JP3145220B2 (de)
AT (1) ATE134611T1 (de)
CA (1) CA2086654C (de)
DE (3) DE4200259A1 (de)
DK (1) DK0554543T3 (de)
ES (1) ES2084914T3 (de)
GR (1) GR3019653T3 (de)
LU (1) LU91869I2 (de)
MX (1) MX9300014A (de)
SG (1) SG48046A1 (de)
ZA (1) ZA9311B (de)

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JP2008538573A (ja) * 2005-04-22 2008-10-30 ワイス ベンゾフラニルアルカナミン誘導体およびその5−ht2cアゴニストとしての使用
AU2006239920A1 (en) * 2005-04-22 2006-11-02 Wyeth Dihydrobenzofuran derivatives and uses thereof
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Also Published As

Publication number Publication date
ATE134611T1 (de) 1996-03-15
CA2086654C (en) 2003-09-23
JP3145220B2 (ja) 2001-03-12
US5384330A (en) 1995-01-24
CA2086654A1 (en) 1993-07-09
EP0554543B1 (de) 1996-02-28
DK0554543T3 (da) 1996-03-18
DE59205496D1 (de) 1996-04-04
EP0554543A3 (en) 1993-10-27
SG48046A1 (en) 1998-04-17
ZA9311B (en) 1993-08-05
ES2084914T3 (es) 1996-05-16
LU91869I2 (fr) 2011-11-14
JPH05345752A (ja) 1993-12-27
DE4200259A1 (de) 1993-07-15
GR3019653T3 (en) 1996-07-31
MX9300014A (es) 1993-07-01
EP0554543A2 (de) 1993-08-11

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