DE60007127D1 - N-pyrazol a2a rezeptor agonisten - Google Patents
N-pyrazol a2a rezeptor agonistenInfo
- Publication number
- DE60007127D1 DE60007127D1 DE60007127T DE60007127T DE60007127D1 DE 60007127 D1 DE60007127 D1 DE 60007127D1 DE 60007127 T DE60007127 T DE 60007127T DE 60007127 T DE60007127 T DE 60007127T DE 60007127 D1 DE60007127 D1 DE 60007127D1
- Authority
- DE
- Germany
- Prior art keywords
- pyrazole
- receptor agonists
- agonists
- receptor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE122011000010C DE122011000010I1 (de) | 1999-06-22 | 2000-06-21 | N-pyrazol a2a rezeptor agonisten |
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US09/338,185 US6403567B1 (en) | 1999-06-22 | 1999-06-22 | N-pyrazole A2A adenosine receptor agonists |
US338185 | 1999-06-22 | ||
PCT/US2000/040281 WO2000078779A2 (en) | 1999-06-22 | 2000-06-21 | N-pyrazole a2a receptor agonists |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60007127D1 true DE60007127D1 (de) | 2004-01-22 |
DE60007127T2 DE60007127T2 (de) | 2004-09-16 |
Family
ID=23323763
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60007127T Expired - Lifetime DE60007127T2 (de) | 1999-06-22 | 2000-06-21 | N-pyrazol a2a rezeptor agonisten |
DE122011000010C Pending DE122011000010I1 (de) | 1999-06-22 | 2000-06-21 | N-pyrazol a2a rezeptor agonisten |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE122011000010C Pending DE122011000010I1 (de) | 1999-06-22 | 2000-06-21 | N-pyrazol a2a rezeptor agonisten |
Country Status (27)
Country | Link |
---|---|
US (9) | US6403567B1 (de) |
EP (1) | EP1189916B1 (de) |
JP (1) | JP4727880B2 (de) |
KR (1) | KR100463300B1 (de) |
CN (1) | CN1167709C (de) |
AR (1) | AR024441A1 (de) |
AT (1) | ATE256141T1 (de) |
AU (1) | AU760806B2 (de) |
BE (1) | BE2011C004I2 (de) |
BR (1) | BRPI0011856B8 (de) |
CA (1) | CA2377746C (de) |
CY (1) | CY2011002I2 (de) |
DE (2) | DE60007127T2 (de) |
DK (1) | DK1189916T3 (de) |
ES (1) | ES2209974T3 (de) |
FR (1) | FR11C0004I2 (de) |
HK (1) | HK1044952B (de) |
IL (2) | IL147198A0 (de) |
LU (1) | LU91785I2 (de) |
MX (1) | MXPA01013325A (de) |
NO (2) | NO322457B1 (de) |
NZ (1) | NZ516334A (de) |
PT (1) | PT1189916E (de) |
TR (1) | TR200200588T2 (de) |
TW (1) | TWI230161B (de) |
WO (1) | WO2000078779A2 (de) |
ZA (1) | ZA200200301B (de) |
Families Citing this family (69)
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US20030078232A1 (en) * | 2001-08-08 | 2003-04-24 | Elfatih Elzein | Adenosine receptor A3 agonists |
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US8470801B2 (en) * | 2002-07-29 | 2013-06-25 | Gilead Sciences, Inc. | Myocardial perfusion imaging methods and compositions |
US20050020915A1 (en) * | 2002-07-29 | 2005-01-27 | Cv Therapeutics, Inc. | Myocardial perfusion imaging methods and compositions |
EP1524984A1 (de) * | 2002-07-29 | 2005-04-27 | Cv Therapeutics, Inc. | Bildgebende verfahren zur myorcardperfusion unter verwendung von a2a-rezeptor-agonisten |
US6914053B2 (en) | 2002-09-09 | 2005-07-05 | Cv Therapeutics, Inc. | Adenosine A3 receptor agonists |
JP4818127B2 (ja) * | 2004-01-27 | 2011-11-16 | ギリアード・パロ・アルト・インコーポレイテッド | アデノシン受容体作動薬を使用する心筋灌流イメージング方法 |
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ATE531377T1 (de) * | 2004-09-20 | 2011-11-15 | Inotek Pharmaceuticals Corp | Purin-derivate und anwendungsverfahren |
CN101076343A (zh) * | 2004-10-20 | 2007-11-21 | Cv医药有限公司 | A2a腺苷受体激动剂的应用 |
GT200500281A (es) * | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
GB0500785D0 (en) * | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
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US20070183995A1 (en) * | 2006-02-09 | 2007-08-09 | Conopco, Inc., D/B/A Unilever | Compounds useful as agonists of A2A adenosine receptors, cosmetic compositions with A2A agonists and a method for using the same |
GB0607950D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
GB0607944D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
AR060607A1 (es) | 2006-04-21 | 2008-07-02 | Novartis Ag | Derivados de purina,composiciones farmaceuticas que los contienen, metodo de preparacion y usos en enfermedades obstructivas o inflamatorias de las vias respiratorias. |
GB0607951D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
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CN106397442B (zh) * | 2015-07-28 | 2020-03-27 | 国药集团国瑞药业有限公司 | 一种瑞加德松的纯化方法 |
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