DE60126286D1 - Substituierte pyrazole - Google Patents

Substituierte pyrazole

Info

Publication number
DE60126286D1
DE60126286D1 DE60126286T DE60126286T DE60126286D1 DE 60126286 D1 DE60126286 D1 DE 60126286D1 DE 60126286 T DE60126286 T DE 60126286T DE 60126286 T DE60126286 T DE 60126286T DE 60126286 D1 DE60126286 D1 DE 60126286D1
Authority
DE
Germany
Prior art keywords
substituted pyrazole
pyrazole
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60126286T
Other languages
English (en)
Other versions
DE60126286T2 (de
Inventor
Guy Breitenbucher
Hui Cai
P Edwards
A Grice
J Gustin
Haripada Khatuya
P Meduna
A Pio
L Tays
Jianmei Wei
Mary Pat Beavers
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceuticals Inc
Original Assignee
Ortho McNeil Pharmaceutical Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho McNeil Pharmaceutical Inc filed Critical Ortho McNeil Pharmaceutical Inc
Publication of DE60126286D1 publication Critical patent/DE60126286D1/de
Application granted granted Critical
Publication of DE60126286T2 publication Critical patent/DE60126286T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
DE60126286T 2000-08-14 2001-08-10 Substituierte pyrazole Expired - Lifetime DE60126286T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US22513800P 2000-08-14 2000-08-14
US225138P 2000-08-14
PCT/US2001/025289 WO2002014314A2 (en) 2000-08-14 2001-08-10 Substituted pyrazoles
US928122 2001-08-10
US09/928,122 US7309703B2 (en) 2000-08-14 2001-08-10 Substituted pyrazoles

Publications (2)

Publication Number Publication Date
DE60126286D1 true DE60126286D1 (de) 2007-03-15
DE60126286T2 DE60126286T2 (de) 2007-11-15

Family

ID=26919335

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60126286T Expired - Lifetime DE60126286T2 (de) 2000-08-14 2001-08-10 Substituierte pyrazole

Country Status (17)

Country Link
US (9) US7589202B2 (de)
EP (1) EP1309591B1 (de)
JP (1) JP5140225B2 (de)
CN (1) CN1329392C (de)
AR (1) AR035714A1 (de)
AT (1) ATE352552T1 (de)
AU (2) AU2001281255B2 (de)
CA (1) CA2419540A1 (de)
CY (1) CY1106032T1 (de)
DE (1) DE60126286T2 (de)
DK (1) DK1309591T3 (de)
ES (1) ES2281434T3 (de)
HK (1) HK1052509B (de)
MX (1) MXPA03001421A (de)
NZ (1) NZ524193A (de)
PT (1) PT1309591E (de)
WO (1) WO2002014314A2 (de)

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Also Published As

Publication number Publication date
JP2004512272A (ja) 2004-04-22
HK1052509A1 (en) 2003-09-19
US7429591B2 (en) 2008-09-30
CA2419540A1 (en) 2002-02-21
US20020040020A1 (en) 2002-04-04
US20070010530A1 (en) 2007-01-11
NZ524193A (en) 2004-12-24
MXPA03001421A (es) 2004-01-26
AU2001281255B2 (en) 2006-07-20
JP5140225B2 (ja) 2013-02-06
US7452890B2 (en) 2008-11-18
ATE352552T1 (de) 2007-02-15
DE60126286T2 (de) 2007-11-15
US7772236B2 (en) 2010-08-10
PT1309591E (pt) 2007-04-30
US7309703B2 (en) 2007-12-18
US20080300255A1 (en) 2008-12-04
AR035714A1 (es) 2004-07-07
CN1329392C (zh) 2007-08-01
EP1309591B1 (de) 2007-01-24
US7589202B2 (en) 2009-09-15
US20070021437A1 (en) 2007-01-25
EP1309591A2 (de) 2003-05-14
US20070004747A1 (en) 2007-01-04
US20070004738A1 (en) 2007-01-04
US20080293732A1 (en) 2008-11-27
DK1309591T3 (da) 2007-03-26
ES2281434T3 (es) 2007-10-01
CN1468239A (zh) 2004-01-14
US20070004754A1 (en) 2007-01-04
US7417046B2 (en) 2008-08-26
WO2002014314A2 (en) 2002-02-21
HK1052509B (zh) 2007-09-07
US20070004755A1 (en) 2007-01-04
US7388011B2 (en) 2008-06-17
AU8125501A (en) 2002-02-25
CY1106032T1 (el) 2011-04-06
WO2002014314A3 (en) 2002-06-06
US7393850B2 (en) 2008-07-01

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