DE60336732D1 - Azaindol-kinaseinhibitoren - Google Patents

Azaindol-kinaseinhibitoren

Info

Publication number
DE60336732D1
DE60336732D1 DE60336732T DE60336732T DE60336732D1 DE 60336732 D1 DE60336732 D1 DE 60336732D1 DE 60336732 T DE60336732 T DE 60336732T DE 60336732 T DE60336732 T DE 60336732T DE 60336732 D1 DE60336732 D1 DE 60336732D1
Authority
DE
Germany
Prior art keywords
kinase inhibitors
azaindole kinase
azaindole
inhibitors
kinase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60336732T
Other languages
English (en)
Inventor
Rajeev Bhide
Rejean Ruel
Carl Thibeault
Heureux Alexandre L
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of DE60336732D1 publication Critical patent/DE60336732D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
DE60336732T 2002-07-19 2003-07-18 Azaindol-kinaseinhibitoren Expired - Lifetime DE60336732D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39725602P 2002-07-19 2002-07-19
US44721303P 2003-02-13 2003-02-13
PCT/US2003/022554 WO2004009601A1 (en) 2002-07-19 2003-07-18 Azaindole kinase inhibitors

Publications (1)

Publication Number Publication Date
DE60336732D1 true DE60336732D1 (de) 2011-05-26

Family

ID=30773005

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60336732T Expired - Lifetime DE60336732D1 (de) 2002-07-19 2003-07-18 Azaindol-kinaseinhibitoren

Country Status (33)

Country Link
US (6) US6969717B2 (de)
EP (3) EP1534290B1 (de)
JP (2) JP4381978B2 (de)
KR (1) KR100901939B1 (de)
CN (3) CN1315833C (de)
AR (1) AR040500A1 (de)
AT (2) ATE505471T1 (de)
AU (2) AU2003254088B2 (de)
BR (2) BR0312801A (de)
CA (2) CA2492804C (de)
CO (1) CO5680407A2 (de)
CY (1) CY1112628T1 (de)
DE (1) DE60336732D1 (de)
DK (1) DK1534290T3 (de)
ES (1) ES2377963T3 (de)
GE (2) GEP20074124B (de)
HK (1) HK1072545A1 (de)
HR (2) HRP20050058A2 (de)
IL (3) IL166129A0 (de)
IS (2) IS7646A (de)
MX (2) MXPA05000716A (de)
MY (1) MY134848A (de)
NO (2) NO330132B1 (de)
NZ (1) NZ537523A (de)
PE (1) PE20040680A1 (de)
PL (2) PL216663B1 (de)
PT (1) PT1534290E (de)
RS (2) RS20050041A (de)
RU (2) RU2331642C2 (de)
SI (1) SI1534290T1 (de)
TW (1) TWI329112B (de)
UA (1) UA82846C2 (de)
WO (2) WO2004009601A1 (de)

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MXPA05008183A (es) * 2003-02-05 2005-10-05 Bristol Myers Squibb Co Proceso para preparar pirrolotriazina como inhibidores de cinasa.

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JP2005538989A (ja) 2005-12-22
EP1539763A4 (de) 2007-08-01
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IS2880B (is) 2014-05-15
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AR040500A1 (es) 2005-04-06
CN1681508B (zh) 2010-10-06
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US20090170853A1 (en) 2009-07-02
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